Quick Facts
What is Tesamorelin?
Tesamorelin is a synthetic analog of human GHRH that contains all 44 amino acids plus a trans-3-hexenoic acid modification that improves stability. It is FDA-approved (as Egrifta) for the treatment of lipodystrophy in HIV patients, making it one of the few peptides with full regulatory approval. Research has demonstrated significant reductions in visceral adipose tissue with its use.
How Does Tesamorelin Work?
Tesamorelin binds to GHRH receptors on the pituitary gland with similar affinity to natural GHRH. The trans-3-hexenoic acid modification at the N-terminus increases its resistance to enzymatic degradation while preserving full biological activity. By stimulating GH release, it indirectly elevates IGF-1 levels, which contributes to its metabolic effects including reduction of visceral fat.
Research-Backed Benefits
Visceral Fat Reduction
Strong EvidenceFDA-approved for reducing trunk fat accumulation with clinically proven efficacy.
Metabolic Improvement
Strong EvidenceMay improve triglyceride levels and other metabolic markers.
Cognitive Function
Moderate EvidenceResearch suggests potential benefits for cognitive function in older adults.
Natural GH Stimulation
Strong EvidencePromotes physiological GH release while maintaining feedback mechanisms.
Body Composition
Moderate EvidenceMay improve overall body composition beyond just visceral fat.
Dosage Guidelines
Disclaimer: This content is for educational purposes only. Peptides are research compounds not approved by the FDA for human use. Always consult with a qualified healthcare provider.
FDA-approved dosing is 2mg daily subcutaneous injection.
Side Effects & Safety
- Injection site reactions
- Arthralgia (joint pain)
- Peripheral edema
- Paresthesia (tingling)
Frequently Asked Questions
References
- Falutz J, et al. "Tesamorelin for the treatment of lipodystrophy." New England Journal of Medicine, 2007. PMID: 17989381
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